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ACP-5862

Glpbio
Catalog No:GC39541-10mM (in 1mL DMSO) CAS No.:2230757-47-6 MDLNo: Brand:Glpbio purity: 特性: Purpose:ACP-5862 是 Acalabrutinib 的主要活性的,循環(huán)的,吡咯烷開環(huán)代謝產物,對于 Bruton 酪氨酸激酶 (BTK) 的 IC50 為 5.0 nM。Acalabrutinib 是一種口服有效的,選擇性的 BTK 抑制劑,IC50 和 EC50 分別為 3 nM 和 8 nM。DMSO: 250 mg/mL (519.20 mM)
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